Does Neurontin inhibit GABA?

Does Neurontin inhibit GABA? Gabapentin, which is used to treat epilepsy, increases GABA concentrations in the brain. Is gabapentin a GABA agonist or antagonist? The anticonvulsant, antihyperalgesic agent gabapentin is an agonist at brain γ-aminobutyric acid type B receptors negatively coupled to voltage-dependent calcium channels. Does gabapentin potentiate GABA? Interestingly, […]

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